Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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256
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270
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256
Tocris Bioscience™ TL 13-22
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Negative control for TL 13-12
257
Tocris Bioscience™ Janelia Fluor 549, SE
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Yellow dye (Reactive group: NHS ester). Applications: super resolution microscopy e.g. dSTORM & STED, confocal, flow and live cell imaging
258
| Target | Muscarinic Acetylcholine Receptor M5/CHRM5 |
|---|---|
| CAS | 2926782-31-0 |
| Purity | 0.98 |
| Chemical Name or Material | (3R,4S)-rel-1-[(2,3-Dihydro-5-benzofuranyl)sulfonyl]-3-fluoro-4-[[(1-methyl-1H-imidazol-2-yl)thio]methyl]piperidine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C18H22FN3O3S2 |
259
Thermo Scientific Chemicals VE-821, 95%
CAS: 1232410-49-9 Molecular Formula: C18H16N4O3S Molecular Weight (g/mol): 368.41 InChI Key: DUIHHZKTCSNTGM-UHFFFAOYSA-N IUPAC Name: 3-amino-6-(4-methanesulfonylphenyl)-N-phenylpyrazine-2-carboxamide SMILES: CS(=O)(=O)C1=CC=C(C=C1)C1=CN=C(N)C(=N1)C(=O)NC1=CC=CC=C1
| CAS | 1232410-49-9 |
|---|---|
| Molecular Weight (g/mol) | 368.41 |
| SMILES | CS(=O)(=O)C1=CC=C(C=C1)C1=CN=C(N)C(=N1)C(=O)NC1=CC=CC=C1 |
| IUPAC Name | 3-amino-6-(4-methanesulfonylphenyl)-N-phenylpyrazine-2-carboxamide |
| InChI Key | DUIHHZKTCSNTGM-UHFFFAOYSA-N |
| Molecular Formula | C18H16N4O3S |
260
| Target | Voltage-gated Potassium Channel Activators |
|---|---|
| CAS | 339287-36-4 |
| Purity | 0.98 |
| Chemical Name or Material | N-(1,2-Dihydro-5-acenaphthylenyl)-4-fluorobenzamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H14FNO |
261
R&D Systems™ Cy5 Labeled Heparan Sulfate Proteoglycan (Cy5-HSPG)
Used as a substrate to study activity of various heparanases and heparinases and protein heparan sulfate interactions
262
Tocris Bioscience™ Dooku 1
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Reversibly blocks Yoda1 activity; does not affect constitutive Piezo1 activity
| Target | Other Piezo Channel Compounds |
|---|---|
| CAS | 2253744-54-4 |
| Purity | 98% |
| Chemical Name or Material | 2-[(2,6-Dichlorobenzyl)thio)-5-(1 H-pyrrol-2-yl)-1,3,4-oxadiazole |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C13H9Cl2N3OS |
| Formula Weight | 326.2 |
263
| CAS | 53902-12-8 |
|---|---|
| Color | White to Light-yellow to Green |
| Solubility | insoluble in water |
| Physical Form | Crystalline Powder |
| Health Hazard 1 | GHS07: Exclamation mark |
| Chemical Name or Material | Tranilast |
| Recommended Storage | Refrigerator +4°C |
| Merck Index | 9646 |
| Molecular Formula | C18 H17 N O5 |
| Formula Weight | 327.33 |
| Melting Point | 166.2°C to 168.2°C |
264
| Target | Ubiquitin Ligase (E3) Inhibitors |
|---|---|
| Purity | 0.98 |
| Chemical Name or Material | N-((1s,4s)-4-(1H-Benzo[d]imidazol-2-yl)cyclohexyl)-2-(((1H-indol-2-yl)methyl)amino)acetamide dihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H27N5O.2HCl |
265
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Tocris Bioscience™ ML T7
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Tocris Bioscience™ ML T7
Inhibitor of phosphatidylserine/CEACAM1 binding to Tim-3
| Target | CEACAM1/CD66a |
|---|---|
| CAS | 459789-75-4 |
| Purity | 0.98 |
| Chemical Name or Material | 5-(2,4-Dichlorophenyl)-3a,6a-dihydro-3-(4-methylphenyl)spiro[1H-furo[3,4-c]pyrrole-1,2'-[2H]indene]-1',3',4,6(3H,5H)-tetrone |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H17Cl2NO5 |
266
Tocris Bioscience™ JT010
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective TRPA1 channel activator (EC50 = 65 nM)
| CAS | 917562-33-5 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 2-Chloro-N-[4-(4-methoxyphenyl)-2-thiazolyl]-N-(3-methoxypropyl)acetamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C16H19ClN2O3S |
| Formula Weight | 354.85 |
267
| CAS | 41340-25-4 |
|---|---|
| Molecular Formula | C17H21NO3 |
268
Tocris Bioscience™ VH 101 phenol-alkylC6-amine
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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VHL ligand with alkyl linker and terminal amine for onward chemistry
269
Tocris Bioscience™ Janelia Fluor™ 635, Tetrazine
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Red dye (Reactive group: tetrazine). Application: confocal microscopy, super resolution microscopy including dSTORM & STED. Suitable for live cell imaging
270
Tocris Bioscience™ PSEM 89S
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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PSAML141F-GlyR and PSAML141F,Y115F-5-HT3 chimeric ion channel agonist
| Target | Pharmacologically Selective Effector Molecules/PSEM |
|---|---|
| CAS | 1336913-03-1 |
| Purity | 98% |
| Chemical Name or Material | N-(3 S)-1-Azabicyclo[2.2.2 ]oct-3-yl-2,5-dimethoxybenzamide trifluoroacetate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C16H22N2O3.CF3CO2H |
| Formula Weight | 404.38 |